跳至主要内容

Jumping Genes May Play An Important Role in GI Cancers

   Gastrointestinal cancer.webp

     

 Gastrointestinal cancer (GI cancer) refers to malignant conditions of the gastrointestinal tract (GI tract) and accessory organs of digestion, including the esophagus, stomach, biliary system, pancreas, small intestine, large intestine, rectum and anus.  The studies state that a jumping gene may play a critical role in the GI cancer.

 

Medicilon can provide various animal models (including renal failure model, anemia animal model, gastric acid secretion animal model, and gastric ulcer model) to test drug effectiveness according to client needs. We can conduct tests on typical digestive system diseases, including gastric acid secretions, gastric ulcers, and renal failure, using rats as subjects.

        Results of a trio of studies done on human cancer tissue biopsies have added to growing evidence that a so-called jumping gene called LINE-1 is active during the development of many gastrointestinal cancers. The John Hopkins scientists who conducted the studies caution there is no proof that the numerous new “insertions” of these rogue genetic elements in the human genome actually cause cancers, but they say their experiments do suggest that these transposons might one day serve as a marker for early cancer diagnosis.  

        Collectively, the studies focus on insertions of a stretch of DNA, the LINE-1 transposon, that, as its name suggests, can produce copies of itself that hop into new areas of the genome and may interrupt normal DNA sequences. This particular genetic interloper, the investigators say, has been in the human genome for so long that an estimated 17% of it is made up of LINE-1 copies, the vast majority of which are now “rusty hulks” of their former selves, unable to move at all. A few, however, are still mobile. Summaries of two of the studies appeared in Nature Medicine and Genome Research, and a report on the third appears this week in PNAS.  

   
 

        Researchers previously reported cases in which new LINE-1 insertions disabled cancer-fighting genes inside tumors, but no one knew how common it was for jumping genes to play a role in cancer development, says Haig Kazazian, M.D., professor of molecular biology and genetics at the Johns Hopkins University School of Medicine’s McKusick-Nathans Institute for Genetic Medicine, who participated in two of the studies. “A challenge we had to overcome to begin to answer that question was detecting new copies of LINE-1 when the human genome already contains so many. It was like finding a needle in a haystack,” he adds.  

   
 

        After Dr. Kazazian and then-graduate student Adam Ewing devised a method to find LINE-1 insertions using genetic sequencing technology, the two worked with research fellow Szilvia Solyom, Ph.D., and other colleagues to analyze the insertions in several types and stages of gastrointestinal cancer tissues biopsies. They compared the DNA insertions they found in colon, pancreatic, and gastric cancer to those in healthy tissue from the same people.  

   
 

        Results showed that new insertions of the still-mobile LINE-1 transposons tended to occur early in cancer development, Dr. Solyom says. For example, she says, a total of 29 new insertions were found in colon polyps, and 24 new insertions were found in samples from seven patients with pancreatic cancer. Of those, 13 were found in both the primary cancer and metastasized cancer cells, indicating that they had occurred before the tumor metastasized. The group’s findings about the timing of insertions in cancer appear in the Genome Research article.  

   
 

        In the study that appears in Nature Medicine, researchers led by Kathleen Burns, M.D., Ph.D., an associate professor of pathology at Johns Hopkins, homed in on LINE-1 insertions in pancreatic cancers. Using tissues from autopsies of 22 people with pancreatic cancer, they compared insertions in normal tissues, primary tumors, and metastases. Of these, 21 of the cancers had LINE-1 insertions that were not present in the patients’ healthy tissue, notes Dr. Burns, and there tended to be more insertions in the metastasized tumors than in the primary tumors, indicating that the insertions are occurring concurrently with cancer progression.  

   
 

        In the third study, graduate student Tara Doucet in Dr. Kazazian’s laboratory and others examined LINE-1 insertions in esophageal cancer and a condition known as Barrett’s esophagus that is sometimes a precursor to cancer. They found new insertions in some, but not all of both patients whose Barrett’s esophagus had not progressed to cancer after 15 or more years, and patients with both Barrett’s esophagus and cancer.  

   
 

        “The key question is whether these insertions are driving cancer development or whether they are just a byproduct of cancer,” says Dr. Kazazian. To help answer that question, his group hopes to analyze the genomes of individual cells to see whether most insertions seen in cancer cells also crop up in normal cells.  

   
 

        Whatever LINE-1’s role in cancer biology turns out to be, adds Dr. Burns, the fact that the transposons are more active in gastrointestinal cancer cells than in healthy cells could eventually make them a powerful tool for early detection.  

   
 

        We will see if more studies or researches saying that the LINE-1 insertions are suitable to fight for the GI cancer in the future.
 

评论

此博客中的热门博文

What is preclinical testing?

In the process of  preclinical testing  of a compound or biological agent into a drug, the compound involved must go through the testing phase. First, we need to identify potential targets that can treat the disease. Then, a variety of compounds or preparations are screened out. Any compound that has shown potential as a drug for the treatment of this disease needs to be tested for toxicity before clinical testing to reduce the possibility of injury. preclinical testing What is the basis of preclinical testing? According to US Food and Drug Administration (FDA) regulations, a series of tests are required before a new drug is approved for use. In the first stage, basic research determines a hypothetical target for the treatment of a certain disease, and then screens small molecules or biological compounds to discover any substance with the potential to treat the disease. Then, a  preclinical research  phase followed, before which, as described above, the potential toxicity of the compou

Inventory of the three major in vitro pharmacokinetic research methods

  The metabolic properties of a compound are an essential factor in whether or not it can be used as a drug in the clinical setting, so pharmacokinetic studies of newly synthesized compounds are required in drug development. In vitro incubation with liver microsomes, recombinant CYP450 enzyme lines, and in vitro incubation with hepatocytes are some of the more common in vitro drug metabolism methods. 1. In vitro incubation method with liver microsomes The metabolic stability and metabolic phenotypes of candidate compounds in different species of liver microsomes are good predictors of the metabolic properties of compounds in vivo. They are practical tools for evaluating candidate compounds in the pre-development phase of drug development. Liver microsomes include rat liver microsomes, human liver microsomes, canine liver microsomes, monkey liver microsomes, and mouse liver microsomes. In in vitro incubation of the liver, microsomes are the "gold standard" for in vitro d

Novel Parkinson’s Therapies Possible with New Mouse Model

Parkinson's disease (PD) is a neurodegenerative disorder that is marked by the accumulation of the protein, α-synuclein (αS), into clumps known as Lewy bodies, which diminish neural health. Now, researchers from Brigham and Women's Hospital (BWH) report the development of a mouse model to induce PD-like αS aggregation, leading to resting tremor and abnormal movement control. The mouse responds to L-DOPA, similarly to patients with PD. The team's study (“Abrogating Native α-Synuclein Tetramers in Mice Causes a L-DOPA-Responsive Motor Syndrome Closely Resembling Parkinson’s Disease”) on the use of this transgenic mouse model appears in  Neuron . “α-Synuclein (αS) regulates vesicle exocytosis but forms insoluble deposits in PD. Developing disease-modifying therapies requires animal models that reproduce cardinal features of PD. We recently described a previously unrecognized physiological form of αS, α-helical tetramers, and showed that familial PD-causing missense mutati